Substituted-nicotinyl thiourea derivatives bearing pyrimidine moiety: synthesis and biological evaluation

文献类型： 外文期刊

第一作者： Ke, Shaoyong

作者： Ke, Shaoyong;Cao, Xiufang

作者机构：

关键词： Nicotinyl thiourea;PTC;Synthesis;Bioactivity

期刊名称：RESEARCH ON CHEMICAL INTERMEDIATES （ 影响因子：2.914； 五年影响因子：2.32 ）

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收录情况： SCI

摘要： A series of substituted-nicotinyl thiourea derivatives containing pyrimidine ring were synthesized in good to excellent yield using PEG-400 as solid-liquid phase transfer catalyst under ultrasonic irradiation. The structures of all newly synthesized compounds were elucidated and confirmed by IR, (1)H NMR and elemental analysis. The preliminary biological tests show that some of the target compounds present good inhibitory activities against the root and stalk of dicotyledon plants and are safe for monocotyledon plants.

分类号： O62

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