Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives

文献类型： 外文期刊

第一作者： Cui, Zi-Ning

作者： Cui, Zi-Ning;Zhang, Li;Ling, Yun;Yang, Xin-Ling;Shi, Yan-Xia;Li, Bao-Ju;Cui, Zi-Ning;Nishida, Yoshihiro

作者机构：

关键词： 2,5-disubstituted-1,3,4-oxadiazole;5-phenyl-2-furan;fungicidal activity;microwave irradiation;synthesis

期刊名称：JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY （ 影响因子：5.279； 五年影响因子：5.269 ）

ISSN： 0021-8561

年卷期： 2012 年 60 卷 47 期

页码：

收录情况： SCI

摘要： A novel series of 1,3,4-oxadiazole derivatives containing a 5-phenyl-2-furan moiety were synthesized from the intermediates diacylhydrazine 3 and acylhydrazone 5 via an efficient approach under microwave irradiation in good yields. Their structures were characterized by IR, H-1 NMR, and elemental analysis. The antifungal tests indicated that the title compounds showed in vivo fungicidal activity against Botrytis cinerea and Rhizoctonia solanii at 500 mu g/mL obviously. Some tested compounds even had a superiority effect over the commercial fungicides 40% Pyrimethanil SC and 3% Validamycin AS. The activity between the title compound and their precursors diacylhydrazine 3 and acylhydrazone 5 was also compared and discussed.

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