Design, Synthesis and Antifungal/Insecticidal Evaluation of Novel Cinnamide Derivatives

文献类型： 外文期刊

第一作者： Yang, Xiaoli

作者： Yang, Xiaoli;Xu, Yanjun;Qin, Zhaohai;Li, Bo;Wan, Shuqing;Yuan, Huizhu

作者机构：

关键词： cinnamide;beta-phenyl ethylamine;fungicidal activity;insecticidal activity

期刊名称：MOLECULES （ 影响因子：4.411； 五年影响因子：4.587 ）

ISSN： 1420-3049

年卷期： 2011 年 16 卷 11 期

页码：

收录情况： SCI

摘要： Twenty novel cinnamamide derivatives were designed and synthesized using as lead compound pyrimorph, whose morpholine moiety was replaced by beta-phenylethylamine. All the compounds were characterized by their spectroscopic data. The fungicidal and insecticidal activities were also evaluated. The preliminary results showed that all the title compounds had certain fungicidal activities against seven plant pathogens at a concentration of 50 mu g/mL, and compounds 11a and 11l showed inhibition ratios of up to 90% against R. solani. Most of the title compounds exhibited moderate nematicidal activities. In general, the morpholine ring may be replaced by other amines and a chlorine atom in the pyridine ring is helpful to fungicidal activity.

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