Synthesis and Insecticidal Activities of Pyrazole-heterocyclic Diamides

文献类型: 外文期刊

第一作者: Ge Qianjian

作者: Ge Qianjian;Du Xiaohua;Chen Liezhong

作者机构:

关键词: bioactive substructure;diamides;ryanodine receptor activator;synthesis;insecticidal activity

期刊名称:CHINESE JOURNAL OF ORGANIC CHEMISTRY ( 影响因子:1.652; 五年影响因子:1.2 )

ISSN: 0253-2786

年卷期: 2011 年 31 卷 9 期

页码:

收录情况: SCI

摘要: 16 novel pyrazole-heterocyclic diamides were synthesized according to the principle of combination of bioactive substructures, and their structures were characterized by IR, (1)H NMR and HRMS techniques. The crystal structure of 3h was determined by X-ray diffraction analysis. Preliminary bioassays showed that some compounds had lethal activities against Mythimna sepatara and Aphis medicaginis at the dosage of 500 mg/L; some of the compounds had lethal activities against the larvae of Ectropis oblique hypulina Wehrli at the dosage of 100 mg/L, the treated insects appeared to have anti-feeding effect.

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