Novel salicylamide derivatives incorporating neonicotinoid pharmacophore: design, synthesis, characterization, and biological evaluation

文献类型： 外文期刊

第一作者： Ke, Shaoyong

作者： Ke, Shaoyong;Zhang, Zhigang;Long, Tong;Liang, Ying;Yang, Ziwen

作者机构：

关键词： Salicylamide derivatives;Neonicotinoid pharmacophore;Synthesis;Biological activity

期刊名称：MEDICINAL CHEMISTRY RESEARCH （ 影响因子：1.965； 五年影响因子：1.98 ）

ISSN：

年卷期：

页码：

收录情况： SCI

摘要： A series of novel salicylamide derivatives containing neonicotinoid pharmacophore were designed and synthesized via multi-step reactions. These compounds were characterized by satisfied spectrum analyses mainly including ~1H NMR and ESI-MS. The preliminary bioassays indicated that some of target compounds exhibited excellent insecticidal activities against Heliothis armigera and Plutella xylostella at the dosage of 31.25 mug/mL.

分类号： R9

  • 相关文献

[1]Synthesis and Bioactivity of Monocyclic beta-Lactams and 4-Thiazolidinones Derivatives Containing Acridinyl. Mahsud, Liwayidin,Imerhasan, Mukhtar,Mahmud, Muhammad Amin,Helil, Setiwaldi,Liu Huajun. 2014

[2]Synthesis and Biological Activity of a Series of Novel N-Substituted beta-Lactams Derived from Natural Gallic Acid. Ke, Shao-Yong,Cao, Xiu-Fang,Wang, Yun-Shen,Li, Shao-Wei,Chen, Chang-Shui. 2011

[3]Synthesis of E-beta-farnesene analogues containing five-membered azaheterocycles and their biological activity. Ling Yun,Yang Xin-Ling,Chen Fu-Heng,Rui Chang-Hui,Fan Xian-Lin. 2008

[4]Synthesis, Crystal Structure and Biological Activity of N-tert-butyl-N-(4-methyl-1,2,3-thiadiazole)-5-yl-N '-(4-methyl-1,2,3-thiadiazole)-5-formyl-N '-3,5-dichloropyridin-2-yl-diacylhydrazine. Wang Huan,Fu Yi-Feng,Fan Zhi-Jin,Song Hai-Bin,Wu Qing-Jun,Zhang You-Jun,Belskaya, N. P.,Bakulev, V. A.. 2011

[5]Synthesis and Biological Properties of Dihydro-Oxadiazine-Based Heterocyclic Derivatives. Ke, S.,Liang, Y.,Wang, K.,Yang, Z.,Cao, X.. 2011

[6]Synthesis and biological activity of novel benzimidazole derivatives as potential antifungal agents. Zhang, Tao,She, Dongmei,Ning, Jun,Mei, Xiangdong,Li, Yaofa,Pan, Wenliang,Gao, Zhanlin.

[7]Synthesis, Crystal Structure and Biological Activity of 6-Alkyl-7-imino-3-phenyl-2-thioxo-2,3,6,7-tetrahydrothiazolo[4,5-d]pyrimidines. Liang Ying,He Hongwu,Liang Ying. 2009

[8]Microwave-assisted synthesis of benzothiazoleurea derivatives. Chen, Wenbin,Li, Kejian,Xi, Zhen,Wang, Yong.

[9]Rational design and efficient synthesis of a fluorescent-labeled jasmonate. Liu, Songbai,Fu, Yuanqing,Sang, Ruocheng,Wang, Wu-Hong,Dang, Ya-Li.

[10]Spirodiclofen Analogues as Potential Lipid Biosynthesis Inhibitors: A Convenient Synthesis, Biological Evaluation, and Structure-Activity Relationship. Ke, Shaoyong,Sun, Tingting,Zhang, Zhigang,Zhang, Ya-Ni,Liang, Ying,Wang, Kaimei,Yang, Ziwen.

[11]Interactions between Meteorus pulchricornis and Spodoptera exigua multiple nucleopolyhedrovirus. Guo, Hui-Fang,Fang, Ji-Chao,Zhong, Wan-Fang,Liu, Bao-Sheng. 2013

[12]Expression of recombinant myostatin propeptide pPIC9K-Msp plasmid in Pichia pastoris. Du, W.,Liu, M. J.,Du, W.,Xia, J.,Zhang, Y.,Liu, M. J.,Li, H. B.,Yan, X. M.,Zhang, J. S.,Li, N.,Zhou, Z. Y.,Xie, W. Z.. 2015

[13]Secondary Metabolites from the Marine Algal-Derived Endophytic Fungi: Chemical Diversity and Biological Activity. Zhang, Peng,Li, Xin,Wang, Bin-Gui,Zhang, Peng.

[14]Isolation and identification of a novel polysaccharide-peptide complex with antioxidant, anti-proliferative and hypoglycaemic activities from the abalone mushroom. Wong, Jack Ho,Ng, Tzi Bun,Li, Ning,Jiang, Yun,Wang, Chang Rong,Zhang, Ni Ye,Qu, Li Yuan,Lv, Peng Yun,Zhao, Ruili,Shi, Bin,Wang, Yin Ping,Wang, Xiao Ying,Liu, Fang,Li, Le,Fang, Jin Cen,Wen, Ting Yi.

[15]Sequence analysis and heterologous expression of lectin-like gene CMLec3 from the medicinal fungus Cordyceps militaris. Bao, Da Peng,Ma, Yuan Wei,Gong, Ming,Li, Yan,Gao, Ying Nv,Yang, Rui Heng,Mao, Wen Jun,Wang, Ying,Yang, Rui Fang. 2018

[16]Chemical Constituents and Biological Activities of Plants from the Genus Ligustrum. She, Gai-Mei,Gao, Bei-Bei,She, Dong-Mei. 2013

[17]Isolation an antimicrobial action of endophytic fungi from sophora flavescens and effects on microorganism circumstances in soil. He, Lu,Wang, Yong,Xu, Hong Bo,Yu, Na,Liu, Na. 2013

[18]Fabrication, Characterization, and Biological Activity of Avermectin Nano-delivery Systems with Different Particle Sizes. Wang, Anqi,Wang, Yan,Sun, Changjiao,Wang, Chunxin,Cui, Bo,Zhao, Xiang,Zeng, Zhanghua,Yao, Junwei,Yang, Dongsheng,Liu, Guoqiang,Cui, Haixin,Wang, Anqi,Wang, Yan,Sun, Changjiao,Wang, Chunxin,Cui, Bo,Zhao, Xiang,Zeng, Zhanghua,Yao, Junwei,Yang, Dongsheng,Liu, Guoqiang,Cui, Haixin. 2018

[19]Synthesis, Crystal Structure and Biological Activity of Novel Anthranilic Diamides Containing 1,2,3-Thiadiazole. Dong, Wei-Li,Xu, Jun-Ying,Liu, Xing-Hai,Li, Zheng-Ming,Li, Bao-Ju,Shi, Yan-Xia. 2008

[20]PGPR (Plant Growth-Promoting Rhizobacteria) in Mulberry Rhizosphere with the Potential of Soil Fertilizer Pollution Control. Wu, Fan,Zhang, Benfeng,Qiu, Nianquan,Liu, Xunli,Song, Zhen,Zhang, Nan,Guo, Hui,Wu, Fan. 2010

作者其他论文 更多>>

微信小程序