您好,欢迎访问湖北省农业科学院 机构知识库!

Synthesis and Biological Activities of N '-Pyridyl(thiazolyl) Methyloxyphenyl-N-arylacyl Urea Derivatives

文献类型: 外文期刊

作者: Liang Ying 1 ; Zhang Zhigang 1 ; Wei San 1 ; Yang Ziwen 1 ;

作者机构: 1.Hubei Acad Agr Sci, Lab Green Chem & Synth, Hubei Biopesticide Engn Res Ctr, Wuhan 430064, Peoples R China

关键词: benzoylurea;synthesis;insecticidal activity

期刊名称:CHINESE JOURNAL OF ORGANIC CHEMISTRY ( 影响因子:1.652; 五年影响因子:1.2 )

ISSN: 0253-2786

年卷期: 2011 年 31 卷 4 期

页码:

收录情况: SCI

摘要: Eight new N'-pyridyl(thiazolyl) methyloxyphenyl-N-arylacyl urea derivatives were synthesized by the nucleophilic addition reaction of pyridyl(thiazolyl) methyloxy aniline with arylacyl isocyanates. Their structures were confirmed by (1)H NMR, IR spectra and elemental analysis. Preliminary biological tests indicated that these compounds exhibited obvious insecticidal activity, especially, compound 5d showed 100% inhibitory activity against Heliothis armigera and Plutella xylostella at 100 mg/L.

  • 相关文献

[1]Novel ether-functional spiro-tetronic acid derivatives: molecule design, convenient synthesis and biological evaluation. Ke, Shaoyong,Zhang, Zhigang,Zhang, Ya-Ni,Shi, Liqiao,Zhou, Ronghua,Jiang, Aibing,Liang, Ying,Yang, Ziwen.

[2]Oxime Carbamates as Potential Insecticidal Agents: Design, Synthesis and Biological Evaluation. Ke, Shaoyong,Yang, Ziwen,Shi, Liqiao,Liu, Manli,Liang, Ying,Wang, Kaimei,Long, Tong,Jiang, Aibing,Zhang, Zhigang. 2015

[3]Multisubstituted indole-acrylonitrile hybrids as potential cytotoxic agents. Ke, Shaoyong,Yang, Ziwen,Zhang, Zhigang,Liang, Ying,Wang, Kaimei,Liu, Manli,Shi, Liqiao.

[4]Anthranilic acid-based diamides derivatives incorporating aryl-isoxazoline pharmacophore as potential anticancer agents: Design, synthesis and biological evaluation. Shi, Liqiao,Hui, Rui,Wei, Yanhong,Liang, Ying,Yang, Ziwen,Ke, Shaoyong.

[5]Structural diversity-guided convenient construction of functionalized polysubstituted butenolides and lactam derivatives. Ke, Shaoyong,Zhang, Ya-Ni,Shu, Wenming,Zhang, Zhigang,Shi, Liqiao,Liang, Ying,Wang, Kaimei,Yang, Ziwen.

[6]Structural diversity-guided convenient construction of functionalized 4H-1,3,4-oxadiazin-5(6H)-one derivatives. Ke, Shaoyong,Wang, Kaimei,Zhang, Zhigang,Zhang, Ya-Ni,Liang, Ying,Shi, Liqiao,Jiang, Aibing,Yang, Ziwen.

[7]Substituted-nicotinyl thiourea derivatives bearing pyrimidine moiety: synthesis and biological evaluation. Ke, Shaoyong,Cao, Xiufang.

[8]Isolation of a cinnamoyl CoA reductase gene involved in formation of stone cells in pear (Pyrus pyrifolia). Lu, Xiao-Peng,Liu, Yong-Zhong,An, Ji-Cui,Peng, Shu-Ang,Hu, Hong-Ju,Lu, Xiao-Peng,Liu, Yong-Zhong,An, Ji-Cui,Peng, Shu-Ang.

[9]Spirodiclofen Analogues as Potential Lipid Biosynthesis Inhibitors: A Convenient Synthesis, Biological Evaluation, and Structure-Activity Relationship. Ke, Shaoyong,Sun, Tingting,Zhang, Zhigang,Zhang, Ya-Ni,Liang, Ying,Wang, Kaimei,Yang, Ziwen.

[10]Novel cycloalkylthiophene-imine derivatives bearing benzothiazole scaffold: Synthesis, characterization and antiviral activity evaluation. Ke, Shaoyong,Yang, Ziwen,Wang, Kaimei,Liang, Ying,Shi, Liqiao,Wei, Yanhong.

[11]Novel salicylamide derivatives incorporating neonicotinoid pharmacophore: design, synthesis, characterization, and biological evaluation. Ke, Shaoyong,Zhang, Zhigang,Long, Tong,Liang, Ying,Yang, Ziwen.

[12]Synthesis of Novel (E)-alpha-(methoxyimino) Benzeneacetate Derivatives and their Fungicidal Activities. Wang, Xianyou,Chen, Peiyun,Pang, Yanping,Zhao, Zhilei,Wu, Guangchen,Wang, Hua.

[13]Acylhydrazone derivatives as potential anticancer agents: Synthesis, bio-evaluation and mechanism of action. Yu, Xifang,Shi, Liqiao,Ke, Shaoyong.

[14]Discovery of novel isatin-dehydroepiandrosterone conjugates as potential anticancer agents. Ke, Shaoyong,Shi, Liqiao,Yang, Ziwen.

[15]Heterocycle-functional gramine analogues: Solvent- and catalyst-free synthesis and their inhibition activities against cell proliferation. Ke, Shaoyong,Shi, Liqiao,Yang, Qingyu,Liang, Ying,Yang, Ziwen,Cao, Xiufang.

[16]Synthesis, Crystal Structure and Biological Activity of 6-Alkyl-7-imino-3-phenyl-2-thioxo-2,3,6,7-tetrahydrothiazolo[4,5-d]pyrimidines. Liang Ying,He Hongwu,Liang Ying. 2009

[17]Synthesis and Biological Activity of a Series of Novel N-Substituted beta-Lactams Derived from Natural Gallic Acid. Ke, Shao-Yong,Cao, Xiu-Fang,Wang, Yun-Shen,Li, Shao-Wei,Chen, Chang-Shui. 2011

[18]Synthesis, Crystal Structure and Biological Activity of alpha-(5-Chloro-3-trifluoromethyl-1-phenylpyrazol-4-carbonyloxy)-alpha-arylmethyl Phosphonates. Liang Ying,He Haifeng,Yang Ziwen,Liang Ying,He Hongwu,He Haifeng. 2012

[19]Novel amide-type ligand bearing bis-pyridine cores: Synthesis, spectral characterizations and X-ray structure analyses. Ke, Shaoyong. 2016

[20]Progress in the Studies on Synthesis and Biological Properties of Butenolide and Its Derivatives. Cao Xiufang,Sun Tingting,Ke Shaoyong. 2010

作者其他论文 更多>>