您好,欢迎访问湖北省农业科学院 机构知识库!

Synthesis and Biological Activity of a Series of Novel N-Substituted beta-Lactams Derived from Natural Gallic Acid

文献类型: 外文期刊

作者: Cao, Xiu-Fang 2 ; Wang, Yun-Shen 2 ; Li, Shao-Wei 2 ; Chen, Chang-Shui 2 ; Ke, Shao-Yong 1 ;

作者机构: 1.Hubei Acad Agr Sci, Hubei Biopesticide Engn Res Ctr, Wuhan 430064, Peoples R China

2.Huazhong Agr Univ, Coll Sci, Wuhan 430070, Peoples R China

关键词: beta-Lactams;Synthesis;Biological activity

期刊名称:JOURNAL OF THE CHINESE CHEMICAL SOCIETY ( 影响因子:1.967; 五年影响因子:1.639 )

ISSN: 0009-4536

年卷期: 2011 年 58 卷 1 期

页码:

收录情况: SCI

摘要: A series of novel beta-lactams derived from natural gallic acid were conveniently synthesized via classical Staudinger ketene-imine cycloaddition reaction. Their structures were confirmed by satisfactory analytical and spectroscopic methods. The preliminary bioassay showed that some of the target compounds exhibited obvious insecticidal activity against Heliothis armigera at the dosage of 0.2 mg/mL.

  • 相关文献

[1]Spirodiclofen Analogues as Potential Lipid Biosynthesis Inhibitors: A Convenient Synthesis, Biological Evaluation, and Structure-Activity Relationship. Ke, Shaoyong,Sun, Tingting,Zhang, Zhigang,Zhang, Ya-Ni,Liang, Ying,Wang, Kaimei,Yang, Ziwen.

[2]Novel salicylamide derivatives incorporating neonicotinoid pharmacophore: design, synthesis, characterization, and biological evaluation. Ke, Shaoyong,Zhang, Zhigang,Long, Tong,Liang, Ying,Yang, Ziwen.

[3]Synthesis, Crystal Structure and Biological Activity of 6-Alkyl-7-imino-3-phenyl-2-thioxo-2,3,6,7-tetrahydrothiazolo[4,5-d]pyrimidines. Liang Ying,He Hongwu,Liang Ying. 2009

[4]Synthesis and Biological Properties of Dihydro-Oxadiazine-Based Heterocyclic Derivatives. Ke, S.,Liang, Y.,Wang, K.,Yang, Z.,Cao, X.. 2011

[5]SOIL BIOLOGICAL AND BIOCHEMICAL QUALITY OF WHEAT-MAIZE CROPPING SYSTEM IN LONG-TERM FERTILIZER EXPERIMENTS. Qi, Ying-Chun,Hu, Cheng.

[6]PGPR (Plant Growth-Promoting Rhizobacteria) in Mulberry Rhizosphere with the Potential of Soil Fertilizer Pollution Control. Wu, Fan,Zhang, Benfeng,Qiu, Nianquan,Liu, Xunli,Song, Zhen,Zhang, Nan,Guo, Hui,Wu, Fan. 2010

[7]Research Advance of Acylhydrazine Derivatives with Biological Activities. Ke Shaoyong,Sun Tingting,Liang Ying,Yang Ziwen. 2010

[8]Progress in the Studies on Natural Bioactive Pyrrolidine-2,4-diones. Liang Ying,Ke Shaoyong,Wang Kaimei,Yang Ziwen. 2010

[9]Multisubstituted indole-acrylonitrile hybrids as potential cytotoxic agents. Ke, Shaoyong,Yang, Ziwen,Zhang, Zhigang,Liang, Ying,Wang, Kaimei,Liu, Manli,Shi, Liqiao.

[10]Anthranilic acid-based diamides derivatives incorporating aryl-isoxazoline pharmacophore as potential anticancer agents: Design, synthesis and biological evaluation. Shi, Liqiao,Hui, Rui,Wei, Yanhong,Liang, Ying,Yang, Ziwen,Ke, Shaoyong.

[11]Structural diversity-guided convenient construction of functionalized polysubstituted butenolides and lactam derivatives. Ke, Shaoyong,Zhang, Ya-Ni,Shu, Wenming,Zhang, Zhigang,Shi, Liqiao,Liang, Ying,Wang, Kaimei,Yang, Ziwen.

[12]Structural diversity-guided convenient construction of functionalized 4H-1,3,4-oxadiazin-5(6H)-one derivatives. Ke, Shaoyong,Wang, Kaimei,Zhang, Zhigang,Zhang, Ya-Ni,Liang, Ying,Shi, Liqiao,Jiang, Aibing,Yang, Ziwen.

[13]Substituted-nicotinyl thiourea derivatives bearing pyrimidine moiety: synthesis and biological evaluation. Ke, Shaoyong,Cao, Xiufang.

[14]Novel ether-functional spiro-tetronic acid derivatives: molecule design, convenient synthesis and biological evaluation. Ke, Shaoyong,Zhang, Zhigang,Zhang, Ya-Ni,Shi, Liqiao,Zhou, Ronghua,Jiang, Aibing,Liang, Ying,Yang, Ziwen.

[15]Isolation of a cinnamoyl CoA reductase gene involved in formation of stone cells in pear (Pyrus pyrifolia). Lu, Xiao-Peng,Liu, Yong-Zhong,An, Ji-Cui,Peng, Shu-Ang,Hu, Hong-Ju,Lu, Xiao-Peng,Liu, Yong-Zhong,An, Ji-Cui,Peng, Shu-Ang.

[16]Novel cycloalkylthiophene-imine derivatives bearing benzothiazole scaffold: Synthesis, characterization and antiviral activity evaluation. Ke, Shaoyong,Yang, Ziwen,Wang, Kaimei,Liang, Ying,Shi, Liqiao,Wei, Yanhong.

[17]Synthesis of Novel (E)-alpha-(methoxyimino) Benzeneacetate Derivatives and their Fungicidal Activities. Wang, Xianyou,Chen, Peiyun,Pang, Yanping,Zhao, Zhilei,Wu, Guangchen,Wang, Hua.

[18]Acylhydrazone derivatives as potential anticancer agents: Synthesis, bio-evaluation and mechanism of action. Yu, Xifang,Shi, Liqiao,Ke, Shaoyong.

[19]Discovery of novel isatin-dehydroepiandrosterone conjugates as potential anticancer agents. Ke, Shaoyong,Shi, Liqiao,Yang, Ziwen.

[20]Heterocycle-functional gramine analogues: Solvent- and catalyst-free synthesis and their inhibition activities against cell proliferation. Ke, Shaoyong,Shi, Liqiao,Yang, Qingyu,Liang, Ying,Yang, Ziwen,Cao, Xiufang.

作者其他论文 更多>>