科研产出
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1Synthesis, Antifungal Activity, and 3D-QASR of Novel 1,2,3,4-Tetrahydroquinoline Derivatives Containing a Pyrimidine Ether Scaffold as Chitin Synthase Inhibitors
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来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
关键词: 1,2,3,4-tetrahydroquinoline; pyrimidine ether scaffold; antifungal activity; 3D-QSAR; chitin synthase inhibitors
年份:2022
3Rational Design, Synthesis, and Biological Investigations of N-Methylcarbamoylguanidinyl Azamacrolides as a Novel Chitinase Inhibitor
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来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
关键词: chitinase; Argifin; inhibitor; azamacrolide; insecticide
年份:2022
4Design and Optimization of Thioglycosyl-naphthalimides as Efficient Inhibitors Against Human O-GlcNAcase
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来源:FRONTIERS IN CHEMISTRY
关键词: thioglycosyl-naphthalimides; ureido glycosides; beta-N-acetylhexosaminidases; human O-GlcNAcase; inhibitors; molecular docking and MD simulations
年份:2019
5Glycosyl triazoles as novel insect beta-N-acetylhexosaminidase OfHex1 inhibitors: Design, synthesis, molecular docking and MD simulations
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来源:BIOORGANIC & MEDICINAL CHEMISTRY
关键词: beta-N-acetyl-D-hexosaminidase; OfHex1; Glycosyl triazoles; Enzyme inhibitors; Molecular docking; MD simulations
年份:2019
6Discovery of Novel Inhibitors Targeting Human O-GlcNAcase: Docking-Based Virtual Screening, Biological Evaluation, Structural Modification, and Molecular Dynamics Simulation
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来源:JOURNAL OF CHEMICAL INFORMATION AND MODELING
年份:2019
7Rational Design, Synthesis, and Biological Investigations of N-Methylcarbamoylguanidinyl Azamacrolides as a Novel Chitinase Inhibitor
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来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
关键词: chitinase; Argifin; inhibitor; azamacrolide; insecticide
年份:2022
8Structure-Based Virtual Screening of Natural Products and Optimization for the Design and Synthesis of Novel CeCht1 Inhibitors as Nematicide Candidates
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来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
关键词: chitinase; natural product; CeCht1 inhibitors; optimization; nematicidal activity
年份:2022
9Design of Inhibitors Targeting Chitin-Degrading Enzymes by Bioisostere Substitutions and Scaffold Hopping for Selective Control of Ostrinia furnacalis
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来源:JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
关键词: Ostriniafurnacalis; insecticide; chitin-degradingenzymes; scaffold hopping
年份:2024
10A soybean cyst nematode suppresses microbial plant symbionts using a lipochitooligosaccharide-hydrolysing enzyme
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来源:NATURE MICROBIOLOGY
年份:2024